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Targeted Protein Degradation: Design Considerations for PROTAC Development

Nathan L Tran1, Georges A Leconte1, Fleur M Ferguson1,2

  • 1Department of Chemistry and Biochemistry, University of California, La Jolla, San Diego, California, USA.

Current Protocols
|December 5, 2022
PubMed

Keywords:
PROTACcompound optimizationmedicinal chemistryproteolysis-targeting chimeratargeted protein degradation

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