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Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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Identification of Triazolopyridines as Selective α5-GABAA Receptor Negative Allosteric Modulators by a Hybridization

György Szabó1, Benedek Imre Károlyi1, Ágnes Gyöngyvér Vaskó1

  • 1Chemistry Division, Gedeon Richter Plc, P.O. Box 27, Budapest 10H-1475, Hungary.

ACS Chemical Neuroscience
|December 16, 2022
PubMed

Keywords:
CNSSARcognitionpenetrabilityselectivitytriazolopyridinesα5-GABAA receptor NAM

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