Related Experiment Video

Updated: Aug 16, 2025

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

Published on: February 20, 2018

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Pathophysiology and pharmacology of G protein-coupled receptors in the heart

Alyssa Grogan1, Emilio Y Lucero1, Haoran Jiang1

  • 1Department of Medicine, Duke University Medical Center, DUMC 3104, 226 CARL Building, Durham, NC 27710, USA.

Cardiovascular Research
|December 19, 2022
PubMed

Keywords:
Allosteric modulatorsBiased signallingG protein-coupled receptorsHeart failure

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