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Updated: Aug 16, 2025

A Semi-High-Throughput Adaptation of the NADH-Coupled ATPase Assay for Screening Small Molecule Inhibitors
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A Semi-High-Throughput Adaptation of the NADH-Coupled ATPase Assay for Screening Small Molecule Inhibitors

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Isoform selectivities of novel 4-hydroxycoumarin imines as inhibitors of myosin II

Joshua D Smith1, Jhonnathan Brawley2, Kate C Bordenave1

  • 1Department of Pharmacology, University of Nevada, School of Medicine, Reno, NV, 89557-0318, USA.

European Journal of Medicinal Chemistry
|December 21, 2022
PubMed

Keywords:
DockingHomology modelHydroxyquinoline imineMyosin inhibitorSelectivityStructure-activity relationships

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