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Next-Generation Heterocyclic Electrophiles as Small-Molecule Covalent MurA Inhibitors

Péter Ábrányi-Balogh1, Aaron Keeley1, György G Ferenczy1

  • 1Medicinal Chemistry Research Group, Research Centre for Natural Sciences, Magyar tudósok krt 2, H-1117 Budapest, Hungary.

Pharmaceuticals (Basel, Switzerland)
|December 23, 2022
PubMed

Keywords:
MurAcovalent inhibitorcysteine labellingheterocyclic electrophilesquaternization

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