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Updated: Aug 16, 2025

Preparation of N-2-alkoxyvinylsulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines
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Synthesis, ADMET Prediction, and Antitumor Profile of Phenoxyhydrazine- 1,3-thiazoles Derivatives

Lucianna Rabelo Pessoa de Siqueira1,2, Larissa Pelágia de Lima Ferreira1,2, Gevanio Bezerra de Oliveira Filho1

  • 1Laboratory of Planning in Medicinal Chemistry, Department of Pharmaceutical Sciences, Center for Health Sciences, Federal University of Pernambuco, 50740-520, Recife, PE, Brazil.

Current Topics in Medicinal Chemistry
|December 27, 2022
PubMed
Abstract

Keywords:
13-ThiazolesAntitumorBioisosterismCancerDU145MOLT-4

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