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Triazole-fused pyrimidines in target-based anticancer drug discovery

Xing-Jie Dai1, Lei-Peng Xue1, Shi-Kun Ji1

  • 1Key Laboratory of Advanced Drug Preparation Technologies, Ministry of Education, China; State Key Laboratory of Esophageal Cancer Prevention & Treatment, Key Laboratory of Henan Province for Drug Quality and Evaluation, Institute of Drug Discovery and Development, School of Pharmaceutical Sciences, Zhengzhou University, 100 Kexue Avenue, Zhengzhou, 450001, Henan Province, China.

European Journal of Medicinal Chemistry
|February 1, 2023
PubMed

Keywords:
Anticancer targetDrug discoverySARsSmall molecule inhibitorsTriazole-fused pyrimidines

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