P2X7 purinergic receptor: A potential target in heart diseases (Review)

Anfal F Bin Dayel1, Asma S Alonazi1, Tahani K Alshammari1

  • 1Department of Pharmacology and Toxicology, College of Pharmacy, King Saud University, 12371 Riyadh, Kingdom of Saudi Arabia.

Molecular Medicine Reports
|February 17, 2023
PubMed

Insights

The P2X7 purinergic receptor (P2X7R) is implicated in heart diseases. Inhibiting P2X7R shows therapeutic potential for conditions like myocardial infarction, myocarditis, and COVID-19-related heart injury.

Area of Science:

  • Cardiology
  • Molecular Biology
  • Pathology

Background:

  • The P2X7 purinergic receptor (P2X7R) is a cation channel activated by extracellular ATP.
  • P2X7R activation is linked to inflammatory, neurodegenerative, orthopedic diseases, and cancer.
  • Evidence suggests P2X7R plays a significant role in various heart conditions.

Purpose of the Study:

  • To review the role of P2X7R in cardiac dysfunction.
  • To discuss P2X7R as a potential therapeutic target for myocardial diseases.

Main Methods:

  • Literature review of studies investigating P2X7R in cardiovascular diseases.
  • Analysis of P2X7R involvement in myocardial ischemia-reperfusion injury, infarction, myocarditis, and cardiomyopathies.
  • Examination of P2X7R activity in COVID-19 patients and its impact on myocardial injury.

Main Results:

  • P2X7R activation can be protective (alleviating ischemia-reperfusion injury) or detrimental (promoting myocardial infarction and myocarditis).
  • P2X7R contributes to cardiomyopathies (diabetic, dilated, hypertrophic) by inducing hypertrophy, fibrosis, and apoptosis.
  • P2X7R inhibition improves cardiac function post-infarction and reduces inflammation in myocarditis.
  • Hyperactivated P2X7R in COVID-19 may cause severe myocardial injury via specific signaling pathways.

Conclusions:

  • P2X7R has a complex, dual role in heart diseases.
  • Targeting P2X7R inhibition offers a promising therapeutic strategy for managing diverse myocardial pathologies.
  • Further research into P2X7R modulation is warranted for cardiovascular disease treatment.

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