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Updated: Aug 8, 2025

Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors
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Structure-Based Design of Bisubstrate Tetracycline Destructase Inhibitors That Block Flavin Redox Cycling

Emily E Williford1, Caitlin M DeAngelo1, Kevin S Blake2

  • 1Department of Chemistry, Washington University in St. Louis, One Brookings Drive, St. Louis, Missouri 63130, United States.

Journal of Medicinal Chemistry
|March 6, 2023
PubMed

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