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Sulfonyl-PYBOX Ligands Enable Kinetic Resolution of α-Tertiary Azides by CuAAC

Yi Gong1, Cai Wang1, Feng Zhou1

  • 1Shanghai Engineering Research Center of Molecular Therapeutics and New Drug Development, Shanghai Key Laboratory of Green Chemistry and Chemical Processes, School of Chemistry and Molecular Engineering, East China Normal University, 3663 N Zhongshan Road, Shanghai, 200062, China.

Angewandte Chemie (International Ed. in English)
|March 6, 2023
PubMed

Keywords:
AzidesCycloadditionHeterocyclesKinetic Resolution

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