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Optimization of 3-aminotetrahydrothiophene 1,1-dioxides with improved potency and efficacy as non-electrophilic

Jeyun Jo1, Jisu Kim1, Lara Ibrahim2

  • 1College of Pharmacy, Pusan National University, Busan 46241, Republic of Korea.

Bioorganic & Medicinal Chemistry Letters
|April 28, 2023
PubMed

Keywords:
ARE activatorDrug-likenessNRF2Non-electrophilicPGK1 inhibitor

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