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The importance of binding kinetics and drug-target residence time in pharmacology

Kevin E Knockenhauer1, Robert A Copeland1

  • 1Accent Therapeutics, Inc., Lexington, Massachusetts, USA.

British Journal of Pharmacology
|May 9, 2023
PubMed

Keywords:
PK–PD relationshipsbinding kineticsdrug optimizationdrug–target residence time

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