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Updated: Jul 29, 2025

A Direct, Early Stage Guanidinylation Protocol for the Synthesis of Complex Aminoguanidine-containing Natural Products
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Guanidines: Synthesis of Novel Histamine H3R Antagonists with Additional Breast Anticancer Activity and

Marek Staszewski1, Magdalena Iwan2, Tobias Werner3

  • 1Department of Synthesis and Technology of Drugs, Medical University of Lodz, Muszyńskiego 1, 90-151 Łódź, Poland.

Pharmaceuticals (Basel, Switzerland)
|May 27, 2023
PubMed

Keywords:
antagonistbreast cancerguanidineshistamine H3 receptormulti-target directed ligand

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