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Updated: Jul 28, 2025

High-throughput Screening for Small-molecule Modulators of Inward Rectifier Potassium Channels
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Automated Patch Clamp Screening of Amiloride and 5-N,N-Hexamethyleneamiloride Analogs Identifies 6-Iodoamiloride as a

Rocio K Finol-Urdaneta1,2, Jeffrey R McArthur2, Ashraf Aboelela3,4

  • 1Electrophysiology Facility for Cell Phenotyping and Drug Discovery, Wollongong, New South Wales 2522, Australia.

Molecular Pharmaceutics
|June 1, 2023
PubMed

Keywords:
6-iodoamilorideASICASIC inhibitionacid-sensing ion channelamiloridesmall moleculesynchropatch

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