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Quinolone analogues of benzothiazinone: Synthesis, antitubercular structure-activity relationship and ADME profiling

Phelelisiwe S Dube1, Lesetja J Legoabe1, Audrey Jordaan2

  • 1Centre of Excellence for Pharmaceutical Sciences, North-West University, Potchefstroom, 2520, South Africa.

European Journal of Medicinal Chemistry
|June 15, 2023
PubMed

Keywords:
BenzothiazinoneDprE1Mycobacterium tuberculosisNitro compoundsQuinolone

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