Pharmacokinetics and safety of prolonged paracetamol treatment in neonates: An interventional cohort study

Sissel Haslund-Krog1, Jessica M Barry2, Angela K Birnbaum2

  • 1Department of Clinical Pharmacology, Bispebjerg and Frederiksberg University Hospital, Copenhagen NV, Denmark.

Insights

Prolonged paracetamol use in neonates for pain management did not show evidence of liver injury. This study found no significant changes in liver safety markers or metabolism with extended paracetamol administration.

Area of Science:

  • Neonatal pharmacology
  • Pediatric pain management
  • Drug metabolism and safety

Background:

  • Neonatal pain is a significant concern requiring effective management.
  • Paracetamol (acetaminophen) is commonly used for pain relief in neonates.
  • Data on the safety and pharmacokinetics of prolonged paracetamol use (>72 hours) in this population are limited.

Purpose of the Study:

  • To investigate the pharmacokinetics of paracetamol in neonates receiving prolonged treatment for pain.
  • To assess the safety profile of extended paracetamol administration in neonates, focusing on liver function.
  • To evaluate potential changes in paracetamol metabolism with prolonged use.

Main Methods:

  • A pharmacokinetic study involving 48 neonates receiving oral or intravenous paracetamol for pain.
  • Collection of 126 plasma samples for measurement of paracetamol and its metabolites.
  • Assessment of liver safety markers (alanine aminotransferase, bilirubin) at different time points during treatment.

Main Results:

  • Thirty-eight neonates received paracetamol for over 72 hours, with a median dose of 10.1 mg/kg.
  • No significant differences in liver safety markers were observed between short-term (<72h) and prolonged (>72h) paracetamol use.
  • Pharmacokinetic parameters including volume of distribution, clearance, steady-state concentration, and half-life were estimated for neonates.

Conclusions:

  • Prolonged paracetamol administration in neonates does not appear to induce liver injury.
  • No significant alterations in paracetamol metabolism were detected with extended use.
  • The findings support the safety of carefully monitored, prolonged paracetamol use for neonatal pain management.
Abstract

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