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Isosteric Replacement of Ester Linkage of Lysophospholipids with Heteroaromatic Rings Retains Potency and Subtype

Masaya Ikubo1, Akiharu Uwamizu2, Luying Chen1

  • 1Department of Organic and Medicinal Chemistry, Graduate School of Pharmaceutical Sciences, The University of Tokyo.

Chemical & Pharmaceutical Bulletin
|July 2, 2023
PubMed

Keywords:
bioisosteric replacementester linkageheteroaromatic ringlysophosphatidylserine (LysoPS)metabolic stability

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