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Updated: Jul 20, 2025

Solid-phase Synthesis of [4.4] Spirocyclic Oximes
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Synthesis of raloxifene-like quinoxaline derivatives by intramolecular electrophilic cyclization with disulfides

Yuhi Umezu1, Eito Horiyama1, Yuto Nakai1

  • 1Department of Chemistry and Biomolecular Science, Faculty of Engineering, Gifu University, 1-1 Yanagido, Gifu 501-1193, Japan.

Bioorganic & Medicinal Chemistry Letters
|August 2, 2023
PubMed

Keywords:
DisulfideHL-60Intramolecular electrophilic cyclizationSK-BR-3Thieno[2,3–b]quinoxaline

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