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Updated: Jul 19, 2025

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Discovery of novel methionine adenosyltransferase 2A (MAT2A) allosteric inhibitors by structure-based virtual

Tuomo Kalliokoski1, Henna Kettunen2, Esa Kumpulainen1

  • 1Orion Pharma, Orionintie 1A, 02101 Espoo, Finland.

Bioorganic & Medicinal Chemistry Letters
|August 17, 2023
PubMed

Keywords:
Allosteric inhibitorMethionine adenosyltransferase 2A (MAT2A)Methylthioadenosine phosphorylase (MTAP)Structure-based virtual screening

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