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A Fluorogenic Peptide Cleavage Assay to Screen for Proteolytic Activity: Applications for coronavirus spike protein activation
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Structure and function of SARS-CoV and SARS-CoV-2 main proteases and their inhibition: A comprehensive review

Xin Li1, Yongcheng Song1

  • 1Department of Pharmacology and Chemical Biology, Baylor College of Medicine, 1 Baylor Plaza, Houston, TX, 77030, USA; Dan L. Duncan Comprehensive Cancer Center, Baylor College of Medicine, 1 Baylor Plaza, Houston, TX, 77030, USA.

European Journal of Medicinal Chemistry
|September 2, 2023
PubMed

Keywords:
Drug discoveryMain proteaseSARS-CoV-2Small-molecule inhibitor

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