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Measuring G-protein-coupled Receptor Signaling via Radio-labeled GTP Binding
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An inverse agonist of orphan receptor GPR61 acts by a G protein-competitive allosteric mechanism

Joshua A Lees1, João M Dias1, Francis Rajamohan1

  • 1Discovery Sciences, Medicine Design, Pfizer Inc., Groton, CT, USA.

Nature Communications
|September 23, 2023
PubMed

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