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Updated: Jul 15, 2025

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission

Published on: August 16, 2018

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Structure-function Studies of GABA (A) Receptors and Related computer-aided Studies

Fatin H Mohamad1, Muhamad Arif Mohamad Jamali2, Ahmad Tarmizi Che Has3

  • 1Department of Neurosciences, School of Medical Sciences, Universiti Sains Malaysia, Health Campus, Kubang Kerian, 16150 Kota Bharu, Kelantan, Malaysia.

Journal of Molecular Neuroscience : MN
|September 26, 2023
PubMed
Summary

The γ-aminobutyric acid type A (GABA) receptor is a complex pentameric protein. Computational studies enhance understanding of GABA receptor structure and function for drug development.

Keywords:
GABA (A) receptorsand benzodiazepinesin silicostructure-function

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