Calcipotriol suppresses GPX4-mediated ferroptosis in OA chondrocytes by blocking the TGF-β1 pathway

Zhicheng Yang1, Wei Jiang2, Chenwei Xiong3

  • 1Department of Orthopedics, The Affiliated Changzhou Second People's Hospital of Nanjing Medical University, China; Changzhou Medical Center, Nanjing Medical University, Changzhou, 213000, China.

Cytokine
|October 2, 2023
PubMed

Insights

Calcipotriol treatment inhibits chondrocyte ferroptosis, a key process in osteoarthritis (OA) progression. This study reveals calcipotriol suppresses the TGF-β1 pathway, offering a new therapeutic avenue for OA joint degeneration.

Area of Science:

  • Biomedical Sciences
  • Molecular Biology
  • Orthopedics

Background:

  • Osteoarthritis (OA) affects millions globally, characterized by joint inflammation and cartilage breakdown.
  • Current OA treatments lack a definitive cure, necessitating research into novel therapeutic mechanisms.
  • Chondrocyte ferroptosis, a form of regulated cell death, is implicated in OA pathogenesis.

Purpose of the Study:

  • To elucidate the molecular mechanisms by which calcipotriol alleviates chondrocyte ferroptosis in osteoarthritis.
  • To investigate the effect of calcipotriol on reactive oxygen species and lipid peroxidation in chondrocytes.
  • To evaluate the therapeutic potential of calcipotriol in an in vivo rat model of osteoarthritis.

Main Methods:

  • Utilized western blotting, qPCR, and immunofluorescence to analyze molecular pathways.
  • Assessed oxidative stress markers using dihydroethidium staining and BODIPY.
  • Employed a destabilized medial meniscus model in rats, followed by intra-articular calcipotriol injection and histological analysis (H&E, Safranin O-Fast Green, micro-CT, IHC).

Main Results:

  • Calcipotriol treatment reduced expression of SOX9, col2a1, Aggrecan, MMP13, and ADAMTS5 in IL-1β-stimulated chondrocytes.
  • Calcipotriol inhibited GPX4-mediated ferroptosis by suppressing transforming growth factor-β1 (TGF-β1) expression.
  • Intra-articular calcipotriol injection significantly reduced cartilage degradation in an OA rat model.

Conclusions:

  • Calcipotriol mitigates osteoarthritis by inhibiting GPX4-mediated chondrocyte ferroptosis.
  • The therapeutic effect of calcipotriol is mediated through the suppression of the TGF-β1 signaling pathway.
  • Calcipotriol demonstrates significant potential as a therapeutic agent for osteoarthritis.

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