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Updated: Jul 13, 2025

Synthesis of Antiviral Tetrahydrocarbazole Derivatives by Photochemical and Acid-catalyzed C-H Functionalization via Intermediate Peroxides CHIPS
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Discovery of dihydropyridinone derivative as a covalent EZH2 degrader

Bin Zhou1, Beilei Wang2, Fengming Zou2

  • 1Anhui Province Key Laboratory of Medical Physics and Technology, Institute of Health and Medical Technology, Hefei Institutes of Physical Science, Chinese Academy of Sciences, Hefei, Anhui, 230031, PR China; University of Science and Technology of China, Hefei, Anhui, 230026, PR China.

European Journal of Medicinal Chemistry
|October 12, 2023
PubMed

Keywords:
Covalent inhibitorEZH2 degraderEnhancer of zeste homolog 2H3K27me3

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