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Synthesis, activity, and their relationships of 2,4-diaminonicotinamide derivatives as EGFR inhibitors targeting

Hideaki Kageji1, Takayuki Momose1, Yasuhito Nagamoto1

  • 1R&D Division, Daiichi Sankyo Co., Ltd., 1-2-58 Hiromachi, Shinagawa-ku, Tokyo 140-8710, Japan.

Bioorganic & Medicinal Chemistry Letters
|December 8, 2023
PubMed

Keywords:
C797SDrug discoveryEGFR

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