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Structural mechanism of TRPV5 inhibition by econazole

José J De Jesús-Pérez1, Matthew Gabrielle2, Sumiyya Raheem2

  • 1Department of Systems Pharmacology and Translational Therapeutics, Perelman School of Medicine, University of Pennsylvania, Philadelphia, PA 19104, USA.

Structure (London, England : 1993)
|December 23, 2023
PubMed

Keywords:
ECNTRPTransient receptor potential channelactivation by PI(4,5)P(2)cryo electron microscopycryo-EMgating mechanism inhibitioninhibition by econazole

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