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Synthesis and structure-activity relationships of aryl fluorosulfate-based inhibitors as novel antitubercular agents

Baiyuan Yang1, Paridhi Sukheja1, Bo Qin1

  • 1Calibr, a Division of Scripps Research, La Jolla, CA 92037, USA.

Bioorganic & Medicinal Chemistry Letters
|December 24, 2023
PubMed

Keywords:
Anti-TB activityAryl fluorosulfateMycobacterium tuberculosisPharmacokineticStructure–activity relationship studiesSuFExSulfur (VI) fluoride exchange

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