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Updated: Jul 7, 2025

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

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Development of Highly Potent, G-Protein Pathway Biased, Selective, and Orally Bioavailable GPR84 Agonists

Pinqi Wang1,2, Arun Raja1,2, Vincent B Luscombe3

  • 1Department of Chemistry, University of Oxford, Mansfield Road, Oxford OX1 3TA, U.K.

Journal of Medicinal Chemistry
|December 26, 2023
PubMed

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