GPCR-G protein selectivity revealed by structural pharmacology

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Updated: Jul 7, 2025

G Protein-selective GPCR Conformations Measured Using FRET Sensors in a Live Cell Suspension Fluorometer Assay
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G Protein-selective GPCR Conformations Measured Using FRET Sensors in a Live Cell Suspension Fluorometer Assay

Published on: September 10, 2016

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Sarah M Bernhard1,2, Jianming Han1,2, Tao Che1,2

  • 1Department of Anesthesiology, Washington University School of Medicine, St. Louis, MO, USA.

The FEBS Journal
|December 27, 2023
PubMed

Keywords:
G proteinGPCRbias signalingselectivitystructural pharmacology

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