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Updated: Jul 4, 2025

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

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Fenofibrate Recognition and Gq Protein Coupling Mechanisms of the Human Cannabinoid Receptor CB1

Tianxin Wang1,2, Wenqin Tang3,4,5, Ziyi Zhao3,4,5

  • 1CAS Key Laboratory of Quantitative Engineering Biology, Institute of Synthetic Biology, Shenzhen Institute of Advanced Technology, Chinese Academy of Sciences, Shenzhen, 518055, China.

Advanced Science (Weinheim, Baden-Wurttemberg, Germany)
|February 1, 2024
PubMed

Keywords:
Gq couplingcryo‐electron microscopyfenofibratehuman cannabinoid receptor 1ligand recognition

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