Related Experiment Video

Updated: Jul 2, 2025

Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors
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Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors

Published on: October 26, 2015

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Kinase inhibitor macrocycles: a perspective on limiting conformational flexibility when targeting the kinome with

Baku Acharya1, Debasmita Saha1,2, Daniel Armstrong1

  • 1Department of Pharmaceutical Sciences, College of Pharmacy, University of Arkansas for Medical Sciences Little Rock AR USA BAFrett@uams.edu.

RSC Medicinal Chemistry
|February 23, 2024
PubMed

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