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Updated: Jul 2, 2025

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Exploration of bromodomain ligand-linker conjugation sites for efficient CBP/p300 heterobifunctional degrader

Praveen Kumar Tiwari1, Sai Reddy Doda1, Raghu Vannam1

  • 1Krantz Family Center for Cancer Research, Massachusetts General Hospital, Charlestown, MA, USA; Harvard Medical School, Boston, MA, USA.

Bioorganic & Medicinal Chemistry Letters
|February 26, 2024
PubMed

Keywords:
AcetyltransferaseCBPPROTACTernary complexp300

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