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Potent, selective and reversible hMAO-B inhibition by benzalphthalides: Synthesis, enzymatic and cellular evaluations

Esther Del Olmo1, Bianca Barboza1, Maria Delgado-Esteban2

  • 1Departamento de Ciencias Farmacéuticas: Química Farmacéutica. Facultad de Farmacia. Universidad de Salamanca, CIETUS, IBSAL. Campus Miguel de Unamuno s/n. 37007 Salamanca, Spain.

Bioorganic Chemistry
|March 8, 2024
PubMed

Keywords:
BenzalphthalidesCellular protectionDockingMonoaminoxidase inhibitorsReversibilitySelectivity

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