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Updated: Jun 29, 2025

A High-Throughput Luciferase Assay to Evaluate Proteolysis of the Single-Turnover Protease PCSK9
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Oral PCSK9 Inhibitors

Anandita Agarwala1, Ramsha Asim2, Christie M Ballantyne3

  • 1Center for Cardiovascular Disease Prevention, Cardiovascular Division, Baylor Scott and White Health Heart Hospital Baylor Plano, Plano, TX, USA.

Current Atherosclerosis Reports
|March 27, 2024
PubMed
Abstract

Keywords:
Drug developmentLipid-lowering therapyPCSK9 inhibitors

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