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Updated: Jun 29, 2025

Identification of Transcription Factor Regulators using Medium-Throughput Screening of Arrayed Libraries and a Dual-Luciferase-Based Reporter
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Discovery of YAP1/TAZ pathway inhibitors through phenotypic screening with potent anti-tumor activity via blockade of

Keith Graham1, Philip Lienau2, Benjamin Bader1

  • 1Bayer AG, Pharmaceuticals, Research & Development, Muellerstr. 178, 13353 Berlin, Germany; Nuvisan ICB GmbH, Muellerstr. 178, 13353 Berlin, Germany.

Cell Chemical Biology
|March 27, 2024
PubMed

Keywords:
Rho-GTPaseTEADYAP1/TAZsmall molecule inhibitor

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