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Updated: Jun 29, 2025

Fluorescence-based Monitoring of PAD4 Activity via a Pro-fluorescence Substrate Analog
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Structure-Activity Relationship of PAD4 Inhibitors and Their Role in Tumor Immunotherapy

Yijiang Jia1,2, Renbo Jia1,2, Ayijiang Taledaohan1,2

  • 1Department of Medicinal Chemistry, School of Pharmaceutical Sciences of Capital Medical University, 10 Xi Tou Tiao, You An Men, Beijing 100069, China.

Pharmaceutics
|March 28, 2024
PubMed

Keywords:
PAD4PAD4 inhibitorantitumor immunitycombination therapy strategiesdrug resistancereviewstructure–activity relationship

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