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Updated: Jun 29, 2025

Facile Preparation of 4-Substituted Quinazoline Derivatives
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Proline-derived quinoline formamide compounds as human urate transporter 1 inhibitors with potent uric acid-lowering

Shengnan Li1, Hui Liao2, Lijun Luo1

  • 1Beijing Key Laboratory of Active Substance Discovery and Druggability Evaluation, Institute of Materia Medica, Peking Union Medical College and Chinese Academy of Medical Sciences, 1 Xian Nong Tan Street, Beijing 100050, PR China.

European Journal of Medicinal Chemistry
|March 28, 2024
PubMed

Keywords:
Anti-inflammatory activityDruggabilityHyperuricemiaQuinoline formamidesURAT1

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