Early life phenobarbital exposure dysregulates the hippocampal transcriptome

Seán Quinlan1, Tahiyana Khan1,2, David McFall1,2

  • 1Department of Physiology and Pharmacology, Georgetown University, Washington, DC, United States.

PubMed

Insights

Phenobarbital (PB) causes broad gene expression changes in neonatal brains, unlike levetiracetam (LEV). This transcriptomic alteration in developing brains may explain PB

Area of Science:

  • Neuroscience
  • Developmental Biology
  • Pharmacology

Background:

  • Phenobarbital (PB) and levetiracetam (LEV) are first-line neonatal seizure treatments.
  • Concerns exist regarding PB's potential for lasting neurodevelopmental toxicity.
  • The impact of these drugs on the neonatal brain's transcriptomic landscape is not fully understood.

Purpose of the Study:

  • To investigate the effects of PB and LEV on the neonatal rat hippocampal transcriptome.
  • To compare the transcriptomic changes induced by PB and LEV exposure during critical neurodevelopmental windows.

Main Methods:

  • Neonatal rat pups received a single dose of PB, LEV, or vehicle.
  • Hippocampal RNA sequencing was performed 72 hours post-administration.
  • Differential gene expression analysis was conducted to identify transcriptomic alterations.

Main Results:

  • PB exposure resulted in 124 differentially expressed transcripts, while LEV exposure affected only 15 transcripts.
  • PB significantly decreased GABAergic and oligodendrocyte markers (pvalb, opalin).
  • PB exposure increased markers of microglial activation (cd68) and astrocyte activity (vegfa).

Conclusions:

  • PB induces widespread transcriptomic changes in the developing brain, suggesting a link to neurotoxicity.
  • LEV appears to have a minimal impact on the neonatal transcriptome compared to PB.
  • These findings highlight PB's potential to disrupt multiple cell types and molecular pathways during critical neurodevelopmental periods.

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