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Updated: Jun 28, 2025

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

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Structure-activity relationship studies of tetrahydroquinolone derivatives as GPR41 modulators

Shinsuke Inuki1, Junki Miyamoto2, Naoki Hashimoto1

  • 1Department of Bioorganic Medicinal Chemistry, Graduate School of Pharmaceutical Sciences, Kyoto University, Sakyo-ku, Kyoto 606-8501, Japan.

Bioorganic & Medicinal Chemistry Letters
|April 19, 2024
PubMed

Keywords:
GPR41Structure–activity relationshipsTetrahydroquinolone

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