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Updated: Jun 28, 2025

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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Application of covalent modality in proximity-induced drug pharmacology: Early development, current strategy, and

Linjie Li1, Song Liu1, Youfu Luo1

  • 1State Key Laboratory of Biotherapy and Cancer Center, West China Hospital, West China Medical School, Sichuan University, Chengdu, 610041, China.

European Journal of Medicinal Chemistry
|April 21, 2024
PubMed

Keywords:
Bi-functional moleculeCovalent moleculePROTACProximity-induced drug

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