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Updated: Jun 26, 2025

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The Benzoylpiperidine Fragment as a Privileged Structure in Medicinal Chemistry: A Comprehensive Review

Giulia Bononi1, Chiara Lonzi1, Tiziano Tuccinardi1

  • 1Department of Pharmacy, University of Pisa, Via Bonanno 6, 56126 Pisa, Italy.

Molecules (Basel, Switzerland)
|May 11, 2024
PubMed

Keywords:
benzoylpiperidinebenzoylpiperidine-based small moleculesbioisosterediagnostic agentsdrug designmedicinal chemistryphenyl(piperidin-4-yl)methanoneprivileged structuretherapeutic agents

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