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Updated: Jun 26, 2025

Radiosynthesis of 1-2-[18F]Fluoroethyl-L-Tryptophan using a One-pot, Two-step Protocol
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Radiosynthesis of 1-2-[18F]Fluoroethyl-L-Tryptophan using a One-pot, Two-step Protocol

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α-Fluorination of tropane compounds and its impact on physicochemical and ADME properties

Tamaki Hoshikawa1, Toshiki Kurokawa1, Hikaru Yoshimura1

  • 1Tsukuba Research Laboratories, Eisai Co., Ltd., Ibaraki, Japan.

Bioorganic & Medicinal Chemistry Letters
|May 16, 2024
PubMed

Keywords:
C-H functionalizationElectrochemistryFluorination

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