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Discovery of first-in-class highly selective TRPV1 antagonists with dual analgesic and hypoglycemic effects

Chunxia Liu1, Wenxin Wang2, Shiyu Zhao1

  • 1Department of Pharmacy, The First Affiliated Hospital of Zhengzhou University, Zhengzhou 450052, PR China; Henan Key Laboratory of Precision Clinical Pharmacy, The First Affiliated Hospital of Zhengzhou University, Zhengzhou 450052, PR China.

Bioorganic & Medicinal Chemistry
|May 22, 2024
PubMed

Keywords:
AnalgesicAntagonistsBlood glucoseFlavonoidsTRPV1

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