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Updated: Jun 13, 2025

Continuous Fluorescence-Based Endonuclease-Coupled DNA Methylation Assay to Screen for DNA Methyltransferase Inhibitors
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Targeting the Tumor Epigenetic Regulator SETDB1 for Tumor Therapy

Cheng Peng1, Nini Zhou1, Tengjiang Chen1

  • 1School of life Sciences, Southwest University, No.2 Tiansheng Road., Beibei, Chongqing, China.

Current Cancer Drug Targets
|September 10, 2024
PubMed
Abstract

Keywords:
Epigenetic modificationcancer progressionhistone methyltransferase SETDB1inhibitorsignal pathwaystumor therapy.

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