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Updated: Jun 11, 2025

Yeast Luminometric and Xenopus Oocyte Electrophysiological Examinations of the Molecular Mechanosensitivity of TRPV4
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Inhibition of TRPV1 by an antagonist in clinical trials is dependent on cholesterol binding

Tal Brandwine-Shemmer1, Baruch Minke1, Irena Levitan2

  • 1Department of Medical Neurobiology, Institute for Medical Research Israel-Canada (IMRIC), Edmond and Lily Safra Center for Brain Sciences (ELSC), Faculty of Medicine, The Hebrew University, Jerusalem, Israel.

Cell Calcium
|October 2, 2024
PubMed

Keywords:
CholesterolLibvatrepTRPV antagonistsTRPV channel

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