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Updated: Jun 9, 2025

An Efficient Method for the Synthesis of Peptoids with Mixed Lysine-type/Arginine-type Monomers and Evaluation of Their Anti-leishmanial Activity
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An Efficient Method for the Synthesis of Peptoids with Mixed Lysine-type/Arginine-type Monomers and Evaluation of Their Anti-leishmanial Activity

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Synthesis and biological evaluation of 4,7,9-trisubstituted benzoxazepines as antileishmanial agents

Tara Man Kadayat1, Stefan Kwiatkowski1, Diana Ortiz2

  • 1Department of Pharmaceutical Sciences, College of Pharmacy, University of Kentucky, Lexington, KY 40536-0509 USA.

Bioorganic & Medicinal Chemistry Letters
|October 30, 2024
PubMed

Keywords:
Antileishmanial agents, Neglected tropical diseaseBenzoxazepineLeishmaniasisPharmacophore analysis

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