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Design and synthesis of indol-2-one derivatives as potential RET inhibitors

Zhenzhu Li1, Kai Sun2, Yuanhong Xu1

  • 1Shanghai Key Laboratory of New Drug Design, School of Pharmacy, East China University of Science and Technology, 130 Meilong Road, Shanghai 200237, China.

Bioorganic & Medicinal Chemistry Letters
|November 4, 2024
PubMed

Keywords:
Cell proliferationRET kinase inhibitorsStructure-activity relationshipStructure-based optimizationindol-2-one

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