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Towards the design of ligands of the internal pocket TEADs C-terminal domain

Florine Toulotte1, Mathilde Coevoet1, Maxime Liberelle1

  • 1Univ Lille, INSERM, CHU Lille, UMR-S 1172, Lille Neuroscience and Cognition Research Center, F-59000, Lille, France.

European Journal of Medicinal Chemistry
|November 21, 2024
PubMed

Keywords:
Breast cancer proliferation inhibitionHippo pathwayTEAD inhibitionTEAD internal pocket

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