4-Hexylresorcinol Enhances Glut4 Expression and Glucose Homeostasis via AMPK Activation and Histone H3 Acetylation

Xiangguo Che1, Ji-Hyeon Oh2, Yei-Jin Kang2

  • 1Department of Biochemistry and Cell Biology, Cell and Matrix Research Institute, School of Medicine, Kyungpook National University, Daegu 41944, Republic of Korea.

Insights

4-hexylresorcinol (4HR) shows promise as a novel antidiabetic agent. It improves glucose homeostasis by enhancing Glut4 expression via AMPK activation and histone acetylation, beneficial for diabetes treatment.

Area of Science:

  • Biochemistry
  • Pharmacology
  • Endocrinology

Background:

  • Diabetes mellitus is a global health concern requiring novel therapeutic strategies.
  • Understanding molecular mechanisms regulating glucose homeostasis is crucial for effective diabetes management.
  • 4-hexylresorcinol (4HR) is explored for its potential antidiabetic properties.

Purpose of the Study:

  • To investigate 4-hexylresorcinol (4HR) as a potential antidiabetic agent.
  • To assess the effects of 4HR on glucose metabolism, Glut4 expression, AMPK phosphorylation, and histone H3 acetylation in liver cells and diabetic rats.

Main Methods:

  • In vitro studies using Huh7 and HepG2 cells treated with 4HR.
  • Western blotting to quantify Glut4, p-AMPK, and Ac-H3 expression.
  • In vivo studies using streptozotocin (STZ)-induced diabetic rats treated with 4HR.

Main Results:

  • 4HR increased GAPDH activity and glucose uptake in vitro.
  • 4HR elevated Glut4, p-AMPK, and Ac-H3 levels in vitro and in vivo.
  • 4HR treatment in diabetic rats lowered blood glucose, mitigated weight loss, and increased hepatic glycogen storage.

Conclusions:

  • 4HR enhances Glut4 expression by upregulating AMPK activity and histone H3 acetylation.
  • 4HR improves hepatic glucose homeostasis in vitro and in vivo.
  • 4HR demonstrates potential as a therapeutic candidate for diabetes treatment.

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