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Compatibility of furosemide with aminoglycoside admixtures

American Journal of Hospital Pharmacy
|January 1, 1985
PubMed

Insights

Furosemide precipitates when mixed with gentamicin sulfate or netilmicin sulfate in intravenous admixtures. Separate administration or thorough flushing of IV lines is recommended to prevent precipitation and ensure patient safety.

Area of Science:

  • Pharmacology
  • Intravenous Drug Compatibility
  • Clinical Pharmacy

Background:

  • Intravenous admixtures are common in healthcare settings.
  • Ensuring compatibility between co-administered drugs is crucial for patient safety.
  • Furosemide and aminoglycosides are frequently administered intravenously.

Purpose of the Study:

  • To evaluate the compatibility of furosemide with intravenous admixtures containing five different aminoglycosides.
  • To identify potential precipitation issues when furosemide is mixed with amikacin, gentamicin, kanamycin, netilmicin, or tobramycin.

Main Methods:

  • Furosemide was added to minibag admixtures of aminoglycosides in dextrose 5% and sodium chloride 0.9%.
  • Visual and microscopic examinations for precipitate were conducted at multiple time points.
  • Simulated Y-site injections were performed, and precipitate analysis included spectrophotometry and melting point determination.

Main Results:

  • Precipitation occurred only when furosemide was added to admixtures containing gentamicin sulfate or netilmicin sulfate.
  • The precipitate was identified as furosemide.
  • Results were consistent in both dextrose 5% and sodium chloride 0.9% solutions and in simulated Y-site injections.

Conclusions:

  • Furosemide is incompatible with gentamicin sulfate and netilmicin sulfate in common intravenous solutions.
  • Separate administration of furosemide or thorough flushing of intravenous lines is necessary when co-administering with these aminoglycosides.
  • This finding is critical for preventing adverse events related to drug precipitation.

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